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Search Results for " neurokinin receptor "

20

Compounds

Cat No. Product Name Synonyms Targets
TP1087 Substance P Neurokinin P Endogenous Metabolite , Neurokinin receptor
Substance P (Neurokinin P) (SP) is an undecapeptide (a peptide composed of a chain of 11 amino acid residues) member of the tachykinin neuropeptide family.
TP1008 Neurokinin A α-Neurokinin,Substance K,Neuromedin L Neurokinin receptor
Neurokinin A (NKA), formerly known as Substance K, is a neurologically active peptide translated from the pre-protachykinin gene.
T7633 Senktide Neurokinin receptor
Senktide is an agonist of tachykinin NK3 receptor.
T23316 SB 218795 Neurokinin receptor
SB 218795 is an effective and selective antagonist of NK3 with a Ki 13 nM for hNK3 which is about 90-fold and 7000-fold selectivity over hNK2 and hNK1.
T16849 SB-222200 Neurokinin receptor
SB-222200 is a selective, reversible, and competitive antagonist of the human NK-3 receptor(Ki=4.4 nM).
TP1086 Men 10376 TFA(135306-85-3,free) Men 10376 TFA,Neurokinin-2 receptor antagonist TFA Neurokinin receptor
Men 10376 TFA(135306-85-3,free) (Neurokinin-2 receptor antagonist TFA) is an effective and selective tachykinin nk-2 receptor antagonist with a K I value of 4.4 M for the nk-2 receptor in the small intestine of rats.
T7209 Maropitant Neurokinin receptor
Maropitant is a selective neurokinin (NK1) receptor antagonist.
TP1572 GR-73632 Neurokinin receptor
Potent and selective tachykinin NK1 receptor agonist (EC50 = 2 nM in guinea pig vas deferens).
T38144 Elinzanetant Neurokinin receptor
Elinzanetant is a dual antagonist of neurokinin (NK) receptors 1 and 3 and modulates reproductive hormone secretion.
T15278 Fezolinetant ESN-364 Neurokinin receptor
Fezolinetant (ESN-364) is an antagonist of the neurokinin 3 receptor (NK3R). It is used for the treatment of menopausal hot flushes.
T7549 Talnetant SB 223412 Neurokinin receptor
Talnetant (SB 223412) is a selective, competitive, brain-penetrant NK3 receptor antagonist with the ability to modulate mesolimbic and mesocortical dopaminergic neurotransmission
T76429 Neurokinin Receptor (393-407), rat
Neurokinin Receptor (393-407), rat (SPR393–407), a fragment of the rat neurokinin 1 receptor (NK1R), undergoes rapid endocytosis and subsequent recycling to the plasma membrane upon substance P (SP) binding. This compoun...
T8235 L-732138 Neurokinin receptor
L-732138 is a potent and competitive antagonist of neurokinin-1 (NK-1) receptor(IC50 : 2.3 nM)
TP1883 [Lys5,MeLeu9,Nle10]-NKA(4-10) Neurokinin receptor
Highy selective and potent NK2 receptor agonist (IC50 = 6.1 nM). Induces contraction of the rat fundus and bladder (EC50 values are 117 and 10 nM respectively).
T17156 Tradipitant VLY-686,LY686017 Neurokinin receptor
Tradipitant (VLY-686) is an antagonist of neurokinin-1.
T7554 Substance P (7-11) Substance P 7-11(TFA) Others , Neurokinin receptor
Substance P (7-11) (Substance P 7-11(TFA)) is a C-terminal fragment of Substance P .
T16038 Men 10376 Neurokinin-2 receptor antagonist CDK
Men 10376 is a selective antagonist of tachykinin NK-2 receptor. It has a Ki of 4.4 μM for rat small intestine NK-2 receptor.
T6905 Netupitant Ro 67-31898/000,CID 6451149 Neurokinin receptor
Netupitant (CID 6451149) is a specific neurokinin 1 (NK1) receptor antagonist (Ki: 0.95 nM).
T3716 Rolapitant SCH619734 Neurokinin receptor
Rolapitant (SCH619734) Hydrochloride is the hydrochloride salt form of rolapitant, an orally bioavailable, centrally-acting, selective, neurokinin 1 receptor (NK1-receptor) antagonist with potential antiemetic activity. ...
T7559 Neurokinin A(4-10) Neurokinin A(4-10)(TFA) Neurokinin receptor
Neurokinin A(4-10)(TFA) is an agonist of tachykinin NK2 receptor .
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TargetMol